Molecular basis for the modulation of resistance to chemotherapeutic agents
Molecular basis for the modulation of resistance to chemotherapeutic agents
Wilhelm Fleischhacker
(ORCID: )
Disciplines
Medical-Theoretical Sciences, Pharmacy (100%)
Keywords
-
Multidrug-Resistenz Modulatoren P-Glykoprotein Struktur-Wirkungs-Beziehungen,
Modulatoren,
Multidrug-Resistenz,
P-Glykoprotein,
Struktur-Wirkungs-Be
Research institution(s)
- Medizinische Universität Wien - 30%
- Universität Wien - 70%
Project participants
- Peter Chiba, Medizinische Universität Wien , associated research partner
- Gerhard F. Ecker, Universität Wien , associated research partner
Research Output
- 228 Citations
- 4 Publications
Publications
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1999
Title Synthesis and in Vitro Multidrug Resistance Modulating Activity of a Series of Dihydrobenzopyrans and Tetrahydroquinolines †DOI 10.1021/jm980517+ Type Journal Article Author Hiessböck R Journal Journal of Medicinal Chemistry Pages 1921-1926 -
1999
Title Structure–activity relationship studies of propafenone analogs based on P-glycoprotein ATPase activity measurements DOI 10.1016/s0006-2952(99)00229-4 Type Journal Article Author Schmid D Journal Biochemical Pharmacology Pages 1447-1456 -
1998
Title Substituted 4-Acylpyrazoles and 4-Acylpyrazolones: Synthesis and Multidrug Resistance-Modulating Activity †DOI 10.1021/jm980121y Type Journal Article Author Chiba P Journal Journal of Medicinal Chemistry Pages 4001-4011 -
1997
Title Studies on Propafenone-type Modulators of Multidrug Resistance III: Variations on the Nitrogen DOI 10.1002/qsar.19970160502 Type Journal Article Author Chiba P Journal Quantitative Structure-Activity Relationships Pages 361-366