Feinabstimmung von 8H-Chinolinen zur Bekämpfung der Krebsres
Fine-tuning 8H-quinolines to target resistance in cancer
Gergely Szakacs
(ORCID: 0000-0002-9311-7827)
Wissenschaftsdisziplinen
Chemie (50%); Medizinisch-theoretische Wissenschaften, Pharmazie (50%)
Keywords
-
Multidrug Resistance,
P-glycoprotein,
Cancer,
Collateral Sensitivity,
Anticancer Chelators,
Solution Speciation
Forschungsstätte(n)
Internationale Projektbeteiligte
- Edit Csapo, University Szegedi - Ungarn
- Istvan Szatmári, University of Szeged - Ungarn
Research Output
- 2 Publikationen
Publikationen
-
2025
Titel Organometallic Half-Sandwich Complexes of 1,10-Phenanthroline Derivatives with Improved Solubility, Albumin-Binding, and Nanoformulation Potential Targeting Drug Resistance in Cancer DOI 10.1021/acs.inorgchem.5c01556 Typ Journal Article Autor Va´Rkonyi E Journal Inorganic Chemistry Seiten 14914-14932 Link Publikation -
2025
Titel Comparative study of multidrug resistance-targeting 8-hydroxyquinoline-amino acid conjugates: anticancer effect, interaction with human serum albumin and organic anion transporting polypeptides DOI 10.1016/j.ejps.2025.107187 Typ Journal Article Autor Dömötör O Journal European Journal of Pharmaceutical Sciences Seiten 107187 Link Publikation